Reaction Details Report a problem with these data
Target
Serine/threonine-protein kinase B-raf [409-765]
Ligand
BDBM185591
Substrate
n/a
Meas. Tech.
RAF Kinase Activity
IC50
56.0±n/a nM
Citation
More Info.:
Target
Name:
Serine/threonine-protein kinase B-raf [409-765]
Synonyms:
B-Raf Protein Kinase | B-Raf proto-oncogene serine/threonine-protein kinase | BRAF | BRAF1 | BRAF_HUMAN | RAFB1 | p94 | v-Raf murine sarcoma viral oncogene homolog B1
Type:
COOH-terminal kinase domain
Mol. Mass.:
40238.92
Organism:
Homo sapiens (Human)
Description:
Recombinant baculoviruses expressing B-RAF (residues 409-765) was purified as a fusion protein.
Residue:
357
Sequence:
SLTNVKALQKSPGPQRERKSSSSSEDRNRMKTLGRRDSSDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSHQFEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPKIHRSASEPSLNRAGFQTEDFSLYACASPKTPIQAGGYGAFPV