Reaction Details
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Target
Cytochrome P450 2A13
Ligand
BDBM84669
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
7.6±0
Temperature
310.15±0 K
IC50
2.1e+3± 1e+2 nM
Citation
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More Info.:
Target
Name:
Cytochrome P450 2A13
Synonyms:
CP2AD_HUMAN | CYP2A13 | CYPIIA13 | Cytochrome P450 2A13 (CYP2A13)
Type:
Protein
Mol. Mass.:
56702.46
Organism:
Homo sapiens (Human)
Description:
Q16696
Residue:
494
Sequence:
MLASGLLLVTLLACLTVMVLMSVWRQRKSRGKLPPGPTPLPFIGNYLQLNTEQMYNSLMKISERYGPVFTIHLGPRRVVVLCGHDAVKEALVDQAEEFSGRGEQATFDWLFKGYGVAFSNGERAKQLRRFSIATLRGFGVGKRGIEERIQEEAGFLIDALRGTHGANIDPTFFLSRTVSNVISSIVFGDRFDYEDKEFLSLLRMMLGSFQFTATSTGQLYEMFSSVMKHLPGPQQQAFKELQGLEDFIAKKVEHNQRTLDPNSPRDFIDSFLIRMQEEEKNPNTEFYLKNLVMTTLNLFFAGTETVSTTLRYGFLLLMKHPEVEAKVHEEIDRVIGKNRQPKFEDRAKMPYTEAVIHEIQRFGDMLPMGLAHRVNKDTKFRDFFLPKGTEVFPMLGSVLRDPRFFSNPRDFNPQHFLDKKGQFKKSDAFVPFSIGKRYCFGEGLARMELFLFFTTIMQNFRFKSPQSPKDIDVSPKHVGFATIPRNYTMSFLPR