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Target
Ecdysone receptor/USP
Ligand
BDBM50178988
Substrate
n/a
Meas. Tech.
ChEMBL_927364 (CHEMBL3072564)
Ki
3.2±n/a nM
Citation
Tohidi-Esfahani, D; Lawrence, MC; Graham, LD; Hannan, GN; Simpson, AM; Hill, RJ Isoforms of the heteropteran Nezara viridula ecdysone receptor: protein characterisation, RH5992 insecticide binding and homology modelling. Pest Manag Sci 67:1457-67 (2011) [PubMed] Article
More Info.:
Target
Name:
Ecdysone receptor/USP
Synonyms:
Ecdysone receptor
Type:
n/a
Mol. Mass.:
n/a
Description:
ASSAY_ID of ChEMBL is 927364
Components:
This complex has 2 components.
Component 1
Name:
Ecdysone receptor
Synonyms:
Ecdysone receptor
Type:
PROTEIN
Mol. Mass.:
61028.87
Organism:
Plodia interpunctella
Description:
ChEMBL_106731
Residue:
541
Sequence:
MRRRWSNNGGFQTLRMLEESSSEVTSSSALGLPPAMVMSPESLASPEYGGLELWSYDDGISYNTATAQLLGNACTMQQQQPPTQPLPSMPLPMPPTTPKSENESMSSGREELSPASSVNGCSTDGDARRQKKGPAPRQQEELCLVCGDRASGYHYNALTCEGCKGFFRRSVTKNAVYIYKFGHACEMDMYMRRKCQECRLKKCLAVGMRPECVVPETQCAIKRKEKKAQREKDKLPVSTTTVDDHMPPIMQCDPPPPEAARIHEVVPRFLSDKLMEQNRLKNIPPLTANQQFLIAGLVWYQDGYEQPSEEDLKRVTQTWQPTDEDDDDMPFRQITEMTILTVQLIVEFAKGLPGFSKISQPDQITLLKACSSEVMMLRVARRYDAATDSVLFANNQAYTRDNYRKAGMAYVIEDLLHFCRCMYSMTMDNVHYALLTAIVIFSDRPGLEQPQLVEEIQRYYLNTLRVYIMNQHSDSPRCAVVFGKILSVLTEIRTLGMQNSNMCISLKLKNRKLPPFLEEIWDVADVSTAQQLPLVDAGSAL
Component 2
Name:
USP
Synonyms:
USP
Type:
PROTEIN
Mol. Mass.:
46808.62
Organism:
Plodia interpunctella
Description:
ChEMBL_106731
Residue:
415
Sequence:
MEPSRESGLNLENSTFMSPMSPPEMKPDTAMLDGLRDDATSPPSFKNYPPNHPLSGSKHLCSICGDRASGKHYGVYSCEGCKGFFKRTVRKDLSYACREERNCIIDKRQRNRCQYCRYQKCLACGMKREAVQEERQRAARGTEDAHPSSSVQVSAEELSIERLLEMEALVADTSEEFQFLRVGPDSNVPPKFRAPVSSLCQIGNKQIAALVVWARDIPHFSQLELEDQVTLIKASWNELLLFAIAWRSMEYLTDERDNVDGSRTTSPPQLMCLMPGMTLHRNSALQAGVGQIFDRVLSELALKMRSLPVDQAEYVALKAVILLNPDVKGLNSRQEVEVLREKMYSCLDEYCRRSRGSEEGRFASLLLRLPALRSISLKSFEHLFFFHLVADGSIPGYIRDALRSHKPPLDASSIM