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Target
Methionine aminopeptidase 2
Ligand
BDBM50531162
Substrate
n/a
Meas. Tech.
ChEMBL_1914456 (CHEMBL4417039)
IC50
14±n/a nM
Citation
Heinrich, T; Seenisamy, J; Becker, F; Blume, B; Bomke, J; Dietz, M; Eckert, U; Friese-Hamim, M; Gunera, J; Hansen, K; Leuthner, B; Musil, D; Pfalzgraf, J; Rohdich, F; Siegl, C; Spuck, D; Wegener, A; Zenke, FT Identification of Methionine Aminopeptidase-2 (MetAP-2) Inhibitor J Med Chem 62:11119-11134 (2019) [PubMed] Article
More Info.:
Target
Name:
Methionine aminopeptidase 2
Synonyms:
Initiation factor 2-associated 67 kDa glycoprotein | MAP 2 | MAP2_HUMAN | METAP2 | MNPEP | MetAP 2 | Methionine aminopeptidase 2 (MetAP2) | Methionine aminopeptidases (HsMetAP2) | P67EIF2 | Peptidase M 2 | p67
Type:
Enzyme
Mol. Mass.:
52884.45
Organism:
Human
Description:
P50579
Residue:
478
Sequence:
MAGVEEVAASGSHLNGDLDPDDREEGAASTAEEAAKKKRRKKKKSKGPSAAGEQEPDKESGASVDEVARQLERSALEDKERDEDDEDGDGDGDGATGKKKKKKKKKRGPKVQTDPPSVPICDLYPNGVFPKGQECEYPPTQDGRTAAWRTTSEEKKALDQASEEIWNDFREAAEAHRQVRKYVMSWIKPGMTMIEICEKLEDCSRKLIKENGLNAGLAFPTGCSLNNCAAHYTPNAGDTTVLQYDDICKIDFGTHISGRIIDCAFTVTFNPKYDTLLKAVKDATNTGIKCAGIDVRLCDVGEAIQEVMESYEVEIDGKTYQVKPIRNLNGHSIGQYRIHAGKTVPIVKGGEATRMEEGEVYAIETFGSTGKGVVHDDMECSHYMKNFDVGHVPIRLPRTKHLLNVINENFGTLAFCRRWLDRLGESKYLMALKNLCDLGIVDPYPPLCDIKGSYTAQFEHTILLRPTCKEVVSRGDDY