Reaction Details Report a problem with these data
Target
Melanocortin receptor 3
Ligand
BDBM50574231
Substrate
n/a
Meas. Tech.
ChEMBL_2122100 (CHEMBL4831247)
Ki
100±n/a nM
Citation
Ericson, MD; Doering, SR; Larson, CM; Freeman, KT; LaVoi, TM; Donow, HM; Santos, RG; Cho, RH; Koerperich, ZM; Giulianotti, MA; Pinilla, C; Houghten, RA; Haskell-Luevano, C Functional Mixture-Based Positional Scan Identifies a Library of Antagonist Tetrapeptide Sequences (LAtTeS) with Nanomolar Potency for the Melanocortin-4 Receptor and Equipotent with the Endogenous AGRP(86-132) Antagonist. J Med Chem 64:14860-14875 (2021) [PubMed] Article
More Info.:
Target
Name:
Melanocortin receptor 3
Synonyms:
MC3-R | MC3R_MOUSE | Mc3r
Type:
PROTEIN
Mol. Mass.:
35808.24
Organism:
Mus musculus
Description:
ChEMBL_1498848
Residue:
323
Sequence:
MNSSCCLSSVSPMLPNLSEHPAAPPASNRSGSGFCEQVFIKPEVFLALGIVSLMENILVILAVVRNGNLHSPMYFFLCSLAAADMLVSLSNSLETIMIAVINSDSLTLEDQFIQHMDNIFDSMICISLVASICNLLAIAIDRYVTIFYALRYHSIMTVRKALTLIGVIWVCCGICGVMFIIYSESKMVIVCLITMFFAMVLLMGTLYIHMFLFARLHVQRIAVLPPAGVVAPQQHSCMKGAVTITILLGVFIFCWAPFFLHLVLIITCPTNPYCICYTAHFNTYLVLIMCNSVIDPLIYAFRSLELRNTFKEILCGCNSMNLG