Reaction Details Report a problem with these data
Target
Adenylate kinase 2, mitochondrial
Ligand
BDBM50367047
Substrate
n/a
Meas. Tech.
ChEMBL_32058 (CHEMBL644156)
Ki
21000000±n/a nM
Citation
Kappler, F; Hai, TT; Abo, M; Hampton, A Species- or isozyme-specific enzyme inhibitors. 8. Synthesis of disubstituted two-substrate condensation products as inhibitors of rat adenylate kinases. J Med Chem 25:1179-84 (1983) [PubMed] Article
More Info.:
Target
Name:
Adenylate kinase 2, mitochondrial
Synonyms:
2.7.4.3 | AK 2 | ATP-AMP transphosphorylase 2 | ATP:AMP phosphotransferase | Adenylate kinase 2 | Adenylate kinase 2, mitochondrial | Adenylate monophosphate kinase | Ak2 | KAD2_RAT
Type:
n/a
Mol. Mass.:
26380.21
Organism:
Rattus norvegicus
Description:
n/a
Residue:
239
Sequence:
MAPNALAPEPEHPEGIRAVLLGPPGAGKGTQAPKLAENFCVCHLATGDMLRAMVASGSELGKKLKATMDAGKLVSDEMVVELIEKNLETPSCKNGFLLDGFPRTVKQAEMLDDLMDKRKEKLDSVIEFSIQDSLLIRRITGRLIHPKSGRSYHEEFNPPKEAMKDDITGEPLIRRSDDNEKALKTRLEAYHTQTTPLVEYYRKRGIHCAIDASQTPDVVFASILAAFSKATCKDLVMFV