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Target
Somatostatin receptor type 4
Ligand
BDBM50369890
Substrate
n/a
Meas. Tech.
ChEMBL_200845 (CHEMBL807055)
Ki
9800±n/a nM
Citation
 Poitout, L; Roubert, P; Contour-Galcéra, MO; Moinet, C; Lannoy, J; Pommier, J; Plas, P; Bigg, D; Thurieau, C Identification of potent non-peptide somatostatin antagonists with sst(3) selectivity. J Med Chem 44:2990-3000 (2001) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4)
Type:
Enzyme
Mol. Mass.:
42015.38
Organism:
Human
Description:
P31391
Residue:
388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCMCPPLPCQQEALQPEPGRKRIPLTRTTTF
  
Inhibitor
Name:
BDBM50369890
Synonyms:
CHEMBL1237140 | CHEMBL1788167
Type:
Small organic molecule
Emp. Form.:
C28H34N4
Mol. Mass.:
426.5964
SMILES:
CCCCC1(CCCC)N[C@@H](Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccccc1 |r|
Structure:
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