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Target
Cathepsin F
Ligand
BDBM50392205
Substrate
n/a
Meas. Tech.
ChEMBL_852645 (CHEMBL2157194)
Ki
>4000±n/a nM
Citation
Frizler, M; Schmitz, J; Schulz-Fincke, AC; Gütschow, M Selective nitrile inhibitors to modulate the proteolytic synergism of cathepsins S and F. J Med Chem 55:5982-6 (2012) [PubMed] Article
More Info.:
Target
Name:
Cathepsin F
Synonyms:
CATF_HUMAN | CATSF | CTSF
Type:
PROTEIN
Mol. Mass.:
53373.38
Organism:
Homo sapiens (Human)
Description:
ChEMBL_852650
Residue:
484
Sequence:
MAPWLQLLSLLGLLPGAVAAPAQPRAASFQAWGPPSPELLAPTRFALEMFNRGRAAGTRAVLGLVRGRVRRAGQGSLYSLEATLEEPPCNDPMVCRLPVSKKTLLCSFQVLDELGRHVLLRKDCGPVDTKVPGAGEPKSAFTQGSAMISSLSQNHPDNRNETFSSVISLLNEDPLSQDLPVKMASIFKNFVITYNRTYESKEEARWRLSVFVNNMVRAQKIQALDRGTAQYGVTKFSDLTEEEFRTIYLNTLLRKEPGNKMKQAKSVGDLAPPEWDWRSKGAVTKVKDQGMCGSCWAFSVTGNVEGQWFLNQGTLLSLSEQELLDCDKMDKACMGGLPSNAYSAIKNLGGLETEDDYSYQGHMQSCNFSAEKAKVYINDSVELSQNEQKLAAWLAKRGPISVAINAFGMQFYRHGISRPLRPLCSPWLIDHAVLLVGYGNRSDVPFWAIKNSWGTDWGEKGYYYLHRGSGACGVNTMASSAVVD