Reaction Details Report a problem with these data
Target
CX3C chemokine receptor 1
Ligand
BDBM50432454
Substrate
n/a
Meas. Tech.
ChEMBL_953474 (CHEMBL2351085)
Ki
220±n/a nM
Citation
Karlström, S; Nordvall, G; Sohn, D; Hettman, A; Turek, D; Åhlin, K; Kers, A; Claesson, M; Slivo, C; Lo-Alfredsson, Y; Petersson, C; Bessidskaia, G; Svensson, PH; Rein, T; Jerning, E; Malmberg, Å; Ahlgen, C; Ray, C; Vares, L; Ivanov, V; Johansson, R Substituted 7-amino-5-thio-thiazolo[4,5-d]pyrimidines as potent and selective antagonists of the fractalkine receptor (CX3CR1). J Med Chem 56:3177-90 (2013) [PubMed] Article
More Info.:
Target
Name:
CX3C chemokine receptor 1
Synonyms:
C-X3-C chemokine receptor 1 | CMKBRL1 | CX3C1_HUMAN | CX3CR1 | GPR13
Type:
PROTEIN
Mol. Mass.:
40399.45
Organism:
Human
Description:
ChEMBL_953474
Residue:
355
Sequence:
MDQFPESVTENFEYDDLAEACYIGDIVVFGTVFLSIFYSVIFAIGLVGNLLVVFALTNSKKPKSVTDIYLLNLALSDLLFVATLPFWTHYLINEKGLHNAMCKFTTAFFFIGFFGSIFFITVISIDRYLAIVLAANSMNNRTVQHGVTISLGVWAAAILVAAPQFMFTKQKENECLGDYPEVLQEIWPVLRNVETNFLGFLLPLLIMSYCYFRIIQTLFSCKNHKKAKAIKLILLVVIVFFLFWTPYNVMIFLETLKLYDFFPSCDMRKDLRLALSVTETVAFSHCCLNPLIYAFAGEKFRRYLYHLYGKCLAVLCGRSVHVDFSSSESQRSRHGSVLSSNFTYHTSDGDALLLL