Reaction Details
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Target
Amiloride-sensitive amine oxidase [copper-containing]
Ligand
BDBM50446752
Substrate
n/a
Meas. Tech.
ChEMBL_1288377 (CHEMBL3118035)
IC50
>1000000±n/a nM
Citation
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More Info.:
Target
Name:
Amiloride-sensitive amine oxidase [copper-containing]
Synonyms:
ABP1 | AOC1 | AOC1_PIG | Amiloride-binding protein 1 | Amine oxidase copper domain-containing protein 1 | DAO | Histaminase | PK-DAO
Type:
PROTEIN
Mol. Mass.:
85480.30
Organism:
Sus scrofa
Description:
ChEMBL_107996
Residue:
755
Sequence:
MGRGTLALGWAGAALLLLQMLAAAERSPRTPGGKAGVFADLSAQELKAVHSFLWSQKELKLEPSGTLTMAKNSVFLIEMLLPKKQHVLKFLDKGHRRPVREARAVIFFGAQEQPNVTEFAVGPLPTPRYMRDLPPRPGHQVSWASRPISKAEYALLSHKLQEATQPLRQFFRRTTGSSFGDCHEQCLTFTDVAPRGLASGQRRTWFILQRQMPGYFLHPTGLELLVDHGSTNAQDWTVEQVWYNGKFYRSPEELAQKYNDGEVDVVILEDPLAKGKDGESLPEPALFSFYQPRGDFAVTMHGPHVVQPQGPRYSLEGNRVMYGGWSFAFRLRSSSGLQILDVHFGGERIAYEVSVQEAVALYGGHTPAGMQTKYIDVGWGLGSVTHELAPDIDCPETATFLDALHHYDADGPVLYPRALCLFEMPTGVPLRRHFNSNFSGGFNFYAGLKGQVLVLRTTSTVYNYDYIWDFIFYPNGVMEAKMHATGYVHATFYTPEGLRYGTRLHTHLIGNMHTHLVNYRVDLDVAGTTNSFQTLQMELENITNPWSPRHRLVQPTLKQTRYSRERQAAFRFGQPLPKYLLITSPKENPWGHTRSYRLQLHSMADQVLPPGWQEERAVTWARYPLAVTRYRESELSSSSIYNQNDPWDPPVVFEEFLRNNENIEDEDLVAWVTVGFLHIPHSEDIPNTATPGNSVGFLLRPFNFFPEDPALASRDLVVVWPLENGSTYAQRWIPEEDQSCLKPPPFSYNGSYRPV