Reaction Details Report a problem with these data
Target
Acrosin
Ligand
BDBM50010124
Substrate
n/a
Meas. Tech.
ChEMBL_1344334 (CHEMBL3257004)
Ki
260±n/a nM
Citation
Parrish, RF; Straus, JW; Paulson, JD; Polakoski, KL; Tidwell, RR; Geratz, JD; Stevens, FM Structure-activity relationships for the inhibition of acrosin by benzamidine derivatives. J Med Chem 21:1132-6 (1979) [PubMed] Article
More Info.:
Target
Name:
Acrosin
Synonyms:
53 kDa fucose-binding protein | ACR | ACRO_PIG | Acrosin heavy chain | Acrosin light chain
Type:
PROTEIN
Mol. Mass.:
45383.66
Organism:
Pig
Description:
ChEMBL_108297
Residue:
415
Sequence:
MLPTAVLLVLAVSVAARDNATCDGPCGLRFRQKLESGMRVVGGMSAEPGAWPWMVSLQIFMYHNNRRYHTCGGILLNSHWVLTAAHCFKNKKKVTDWRLIFGANEVVWGSNKPVKPPLQERFVEEIIIHEKYVSGLEINDIALIKITPPVPCGPFIGPGCLPQFKAGPPRAPQTCWVTGWGYLKEKGPRTSPTLQEARVALIDLELCNSTRWYNGRIRSTNVCAGYPRGKIDTCQGDSGGPLMCRDRAENTFVVVGITSWGVGCARAKRPGVYTSTWPYLNWIASKIGSNALQMVQLGTPPRPSTPAPPVRPPSVQTPVRPPWYFQRPPGPSQQPGSRPRPPAPPPAPPPPPPPPPPPPPPPPPPPQQVSAKPPQALSFAKRLQQLIEALKGTAFSSGRSYYETETTDLQELPAS