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Target
Protein delta homolog 1
Ligand
BDBM50042940
Substrate
n/a
Meas. Tech.
ChEMBL_1444684 (CHEMBL3377246)
Ki
0.400000±n/a nM
Citation
Abdel-Magid, AF Dual leucine zipper kinase inhibitors: potential treatments for neurodegenerative diseases. ACS Med Chem Lett 6:11-2 (2015) [PubMed] Article
More Info.:
Target
Name:
Protein delta homolog 1
Synonyms:
DLK | DLK-1 | DLK1 | DLK1_HUMAN | FA1 | Fetal antigen 1 | pG2
Type:
PROTEIN
Mol. Mass.:
41294.81
Organism:
Human
Description:
ChEMBL_1444684
Residue:
383
Sequence:
MTATEALLRVLLLLLAFGHSTYGAECFPACNPQNGFCEDDNVCRCQPGWQGPLCDQCVTSPGCLHGLCGEPGQCICTDGWDGELCDRDVRACSSAPCANNRTCVSLDDGLYECSCAPGYSGKDCQKKDGPCVINGSPCQHGGTCVDDEGRASHASCLCPPGFSGNFCEIVANSCTPNPCENDGVCTDIGGDFRCRCPAGFIDKTCSRPVTNCASSPCQNGGTCLQHTQVSYECLCKPEFTGLTCVKKRALSPQQVTRLPSGYGLAYRLTPGVHELPVQQPEHRILKVSMKELNKKTPLLTEGQAICFTILGVLTSLVVLGTVGIVFLNKCETWVSNLRYNHMLRKKKNLLLQYNSGEDLAVNIIFPEKIDMTTFSKEAGDEEI