Reaction Details
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Target
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 2
Ligand
BDBM50082117
Substrate
n/a
Meas. Tech.
ChEMBL_1475279 (CHEMBL3425139)
IC50
15±n/a nM
Citation
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More Info.:
Target
Name:
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 2
Synonyms:
6-phosphofructo-2-kinase | 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 2 | 6PF-2-K/Fru-2,6-P2ase 2 | 6PF-2-K/Fru-2,6-P2ase heart-type isozyme | F262_HUMAN | Fructose-2,6-bisphosphatase | PFK/FBPase 2 | PFKFB2
Type:
PROTEIN
Mol. Mass.:
58485.20
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109607
Residue:
505
Sequence:
MSGASSSEQNNNSYETKTPNLRMSEKKCSWASYMTNSPTLIVMIGLPARGKTYVSKKLTRYLNWIGVPTKVFNLGVYRREAVKSYKSYDFFRHDNEEAMKIRKQCALVALEDVKAYLTEENGQIAVFDATNTTRERRDMILNFAEQNSFKVFFVESVCDDPDVIAANILEVKVSSPDYPERNRENVMEDFLKRIECYKVTYRPLDPDNYDKDLSFIKVINVGQRFLVNRVQDYIQSKIVYYLMNIHVQPRTIYLCRHGESEFNLLGKIGGDSGLSVRGKQFAQALRKFLEEQEITDLKVWTSQLKRTIQTAESLGVPYEQWKILNEIDAGVCEEMTYAEIEKRYPEEFALRDQEKYLYRYPGGESYQDLVQRLEPVIMELERQGNVLVISHQAVMRCLLAYFLDKGADELPYLRCPLHTIFKLTPVAYGCKVETIKLNVEAVNTHRDKPTNNFPKNQTPVRMRRNSFTPLSSSNTIRRPRNYSVGSRPLKPLSPLRAQDMQEGAD