Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 2
Ligand
BDBM50015490
Substrate
n/a
Ki
1.8±n/a nM
Comments
PDSP_1370
Citation
Weinberg, DH; Sirinathsinghji, DJ; Tan, CP; Shiao, LL; Morin, N; Rigby, MR; Heavens, RH; Rapoport, DR; Bayne, ML; Cascieri, MA; Strader, CD; Linemeyer, DL; MacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem 271:16435-8 (1996) [PubMed] Article
More Info.:
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY2R_MOUSE | Npy2r | Npy2r protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42634.12
Organism:
Mouse
Description:
P97295
Residue:
381
Sequence:
MGPVGAEADENQTVEVKVEPYGPGHTTPRGELPPDPEPELIDSTKLVEVQVILILAYCSIILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSVYGTVYSLSTLLILYVLPLGIISFSYTRIWSKLRNHVSPGAASDHYHQRRHKMTKMLVCVVVVFAVSWLPLHAFQLAVDIDSHVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSMTFKAKKNLEVKKNNGPTDSFSEATNV
Inhibitor
Name:
BDBM50015490
Synonyms:
CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITRQRY-NH2 | NPY | NPY, human | NPY, human, rat | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly-Glu-Asp-Ala-Pro- Ala-Glu-Asp-Met-Ala-Arg-Tyr-Tyr-Ser-Ala-Leu-Arg-His- Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH2 (NPY) | human Neuropeptide Y
Type:
Small organic molecule
Emp. Form.:
C189H285N55O57S
Mol. Mass.:
4271.685
SMILES:
n/a