Reaction Details Report a problem with these data
Target
Galanin receptor type 2
Ligand
BDBM85073
Substrate
n/a
Ki
28±n/a nM
Comments
PDSP_3166
Citation
 Howard, AD; Tan, C; Shiao, LL; Palyha, OC; McKee, KK; Weinberg, DH; Feighner, SD; Cascieri, MA; Smith, RG; Van Der Ploeg, LH; Sullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett 405:285-90 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 2
Synonyms:
GALR2_RAT | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galnr2 | Galr2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40697.04
Organism:
RAT
Description:
Galanin R2 GALR2 RAT::O08726
Residue:
372
Sequence:
MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIIIVAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPNCTASSRTLDPAC
  
Inhibitor
Name:
BDBM85073
Synonyms:
CAS_3043476 | Galantide (M15) | NSC_3043476
Type:
Small organic molecule
Emp. Form.:
C23H30N2O3
Mol. Mass.:
382.4959
SMILES:
COc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1
Structure:
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