Reaction Details Report a problem with these data
Target
Cholinergic receptor nicotinic alpha 5 subunit
Ligand
BDBM86041
Substrate
n/a
Ki
2.1±n/a nM
Comments
PDSP_2906
Citation
Avalos, M; Parker, MJ; Maddox, FN; Carroll, FI; Luetje, CW Effects of pyridine ring substitutions on affinity, efficacy, and subtype selectivity of neuronal nicotinic receptor agonist epibatidine. J Pharmacol Exp Ther 302:1246-52 (2002) [PubMed] Article
More Info.:
Target
Name:
Cholinergic receptor nicotinic alpha 5 subunit
Synonyms:
Cholinergic, Nicotinic Alpha3Beta4x
Type:
Enzyme Catalytic Domain
Mol. Mass.:
53319.71
Organism:
Xenopus
Description:
Cholinergic, Nicotinic Alpha3Beta4x 0 Xenopus::F7ELS1
Residue:
461
Sequence:
MPWCAEYLLWLFLCLDILHGACGISEPSYIAKSEDRLFKYLFQQQDYQRWVRPVEHLNDTVKVKFGLAITQLVDVDEKNQLMTTNVWLKQEWVDVKLRWDPNEFAGITSIRVPSDSIWIPDIVLYDNADGRFEGSVTKAVVRYDGTINWTPPANYKSSCTIDVTFFPFDLQNCSMKFGSWTYDGSQVDIILEDYHVDKRDFFDNGEWEIVNATGNKGNRTDGCCFYPYITYSFIIKRLPLFYTLFLIIPCIGLSFLTILVFYLPSNEGEKISLCTSVLVSLTVFLLVIEEIIPSSSKVIPLIGEYLVFTMIFVTLSIVLTVFAINIHNRSSATHNAMAPWVRKIFLHKLPKLLCMRSHVDRYFTRKDETGKVRGPESSRNTLEAALDSIRYITRHVMKEHEVQEVVEDWKFVAQVLDRMFLWTFLLVSVIGSLFLFIPVIHKWANIIVPVHIGNMYGDKNT