Reaction Details Report a problem with these data
Target
Cholinergic receptor, nicotinic alpha 1
Ligand
BDBM86040
Substrate
n/a
Ki
0.044±n/a nM
Comments
PDSP_2900
Citation
Avalos, M; Parker, MJ; Maddox, FN; Carroll, FI; Luetje, CW Effects of pyridine ring substitutions on affinity, efficacy, and subtype selectivity of neuronal nicotinic receptor agonist epibatidine. J Pharmacol Exp Ther 302:1246-52 (2002) [PubMed] Article
More Info.:
Target
Name:
Cholinergic receptor, nicotinic alpha 1
Synonyms:
Cholinergic, Nicotinic Alpha4Beta4 | acetylcholine receptor subunit alpha-1-A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52341.78
Organism:
clawed frog
Description:
Cholinergic, Nicotinic Alpha4Beta4 0 Xenopus::F6RLA9
Residue:
457
Sequence:
MDFSLTRLIFLFIAATLVFSSEDESRLINDLFKSYNKVVRPVKAFKDKVVVTLGLQLIQLINVDEVNQIVTTNVRLKQQWEDVHLKWNPEDYGGIKKVRISSGDIWRPDIVLYNNADGDFAIVQETKVLLDYTGKIIWTPPAIFKSYCEMIVTYFPFDLQNCSMKLGTWTYDGSLVVINPESDRPDLSNFMESGEWYMKDYRGWKHWVYYDCCPETPYLDITYHFLLQRLPLYFIVNVVIPCLLFSFLTGLVFYLPTDSGEKITLSVSVLLSLVVFLLVIVELIPSTSSAVPLIGKYMLFTMVFVITSIVITVIVINTHHRSPSTHIMPQWLKKIFIETIPRVMFFSTMKRPAQDQQKKKIFTEDIDISDISGKLGPAAVKYQSPILKNPDVKSAIEGAKYIAETMKSDQESNKASEEWKFVAMVLDHLLLAVFMIVCIIGTLAIFAGRLIELHMQG