Reaction Details Report a problem with these data
Target
Gamma-hydroxybutyrate receptor
Ligand
BDBM86152
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_3053
Citation
Wu, H; Zink, N; Carter, LP; Mehta, AK; Hernandez, RJ; Ticku, MK; Lamb, R; France, CP; Coop, A A tertiary alcohol analog of gamma-hydroxybutyric acid as a specific gamma-hydroxybutyric acid receptor ligand. J Pharmacol Exp Ther 305:675-9 (2003) [PubMed] Article
More Info.:
Target
Name:
Gamma-hydroxybutyrate receptor
Synonyms:
Gamma hydroxybutyric, GHB | Gamma-hydroxybutyrate receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
56171.11
Organism:
RAT
Description:
Gamma hydroxybutyric, GHB 0 RAT::Q6RY99
Residue:
512
Sequence:
MRAAAAGLGPGRLHAWAARRGLGRFPARVPRAAGGRSPCPASISNSRTLRLAAAGNTFCLASTLSSGCWEPCSWPSASGPGVRRAFFPTSQGGQIQGGLDPVWLFVVIGGIMSVLGFAGCIGALRENTFLLKFFSVFLGLIFFLELAAGILAFVFKDWIRDQLNLFINNNVKAYRDDIDLQNLIDFAQEYWSCCGARGPNDWNLNIRTSTALTSNPSRERCGVPFFCWVRTLRKTSQYPCGYTSAQTELEHKIHLHQSWWPFEKWLKKPDGWPGLGAIASFKMGIAGPNPRSTSRQERPTGKLPGVMATCLAHRAVVGASKDALPHSQWQGLWDVCYDLSPRLCEHGTQEATEAGLGLNWGCTGAGLGLFTTELCVWGVHMCVCVCVCVCVRVCLCLCVRVRGMHVCALVSTPGVSTPLLVRWWPFQSFKGDGARRVGHVPASPSLLWDVSLCGLGACCLRPLHIHHDLEPAWSSPWPQCHSLEMGPRILSVSLSRLPLRTHTWQDGYERLN