Reaction Details Report a problem with these data
Target
Kallikrein-14
Ligand
BDBM113299
Substrate
n/a
Meas. Tech.
KLK14 Assay
pH
8±n/a
Temperature
310.15±n/a K
Ki
500±n/a nM
Comments
extracted
Citation
Wagberg, F; Leonardsson, G Benzoxazinone derivatives for treatment of skin diseases US Patent US9695194 Publication Date 7/4/2017
More Info.:
Target
Name:
Kallikrein-14
Synonyms:
KLK-L6 | KLK14 | KLK14_HUMAN | KLKL6 | Kallikrein 14 | Kallikrein-14 | Kallikrein-like protein 6 | hK14
Type:
PROTEIN
Mol. Mass.:
29136.99
Organism:
Human
Description:
ChEMBL_1282452
Residue:
267
Sequence:
MSLRVLGSGTWPSAPKMFLLLTALQVLAIAMTQSQEDENKIIGGHTCTRSSQPWQAALLAGPRRRFLCGGALLSGQWVITAAHCGRPILQVALGKHNLRRWEATQQVLRVVRQVTHPNYNSRTHDNDLMLLQLQQPARIGRAVRPIEVTQACASPGTSCRVSGWGTISSPIARYPASLQCVNINISPDEVCQKAYPRTITPGMVCAGVPQGGKDSCQGDSGGPLVCRGQLQGLVSWGMERCALPGYPGVYTNLCKYRSWIEETMRDK