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Target
Suppressor of tumorigenicity 14 protein [596-855]
Ligand
BDBM236494
Substrate
n/a
Meas. Tech.
Inhibition Enzymatic Assay
pH
7.4±n/a
Temperature
298.15±n/a K
Ki
1.4±0.3 nM
Comments
extracted
Citation
Richter, M; Leduc, R; Colombo, E; Marsault, E Matriptase inhibitors and uses thereof against orthomyxoviridae infections US Patent US9365853 Publication Date 6/14/2016
More Info.:
Target
Name:
Suppressor of tumorigenicity 14 protein [596-855]
Synonyms:
Matriptase | PRSS14 | SNC19 | ST14 | ST14_HUMAN | TADG15
Type:
Enzyme
Mol. Mass.:
28561.29
Organism:
Human
Description:
amino acids 596-855
Residue:
260
Sequence:
GSDEKDCDCGLRSFTRQARVVGGTDADEGEWPWQVSLHALGQGHICGASLISPNWLVSAAHCYIDDRGFRYSDPTQWTAFLGLHDQSQRSAPGVQERRLKRIISHPFFNDFTFDYDIALLELEKPAEYSSMVRPICLPDASHVFPAGKAIWVTGWGHTQYGGTGALILQKGEIRVINQTTCENLLPQQITPRMMCVGFLSGGVDSCQGDSGGPLSSVEADGRIFQAGVVSWGDGCAQRNKPGVYTRLPLFRDWIKENTGV