Reaction Details
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Target
Serine hydroxymethyltransferase, mitochondrial [30-504]
Ligand
BDBM512964
Substrate
n/a
Meas. Tech.
SHMT1 and SHMT2 Activity Assays
IC50
5500±n/a nM
Citation
More Info.:
Target
Name:
Serine hydroxymethyltransferase, mitochondrial [30-504]
Synonyms:
GLYM_HUMAN | SHMT2 | Serine hydroxymethyltransferase, mitochondrial (30-504)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52566.80
Organism:
Homo sapiens (Human)
Description:
aa 30-504
Residue:
475
Sequence:
NAAQTQTGEANRGWTGQESLSDSDPEMWELLQREKDRQCRGLELIASENFCSRAALEALGSCLNNKYSEGYPGKRYYGGAEVVDEIELLCQRRALEAFDLDPAQWGVNVQPYSGSPANLAVYTALLQPHDRIMGLDLPDGGHLTHGYMSDVKRISATSIFFESMPYKLNPKTGLIDYNQLALTARLFRPRLIIAGTSAYARLIDYARMREVCDEVKAHLLADMAHISGLVAAKVIPSPFKHADIVTTTTHKTLRGARSGLIFYRKGVKAVDPKTGREIPYTFEDRINFAVFPSLQGGPHNHAIAAVAVALKQACTPMFREYSLQVLKNARAMADALLERGYSLVSGGTDNHLVLVDLRPKGLDGARAERVLELVSITANKNTCPGDRSAITPGGLRLGAPALTSRQFREDDFRRVVDFIDEGVNIGLEVKSKTAKLQDFKSFLLKDSETSQRLANLRQRVEQFARAFPMPGFDEH