Reaction Details
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Target
Glucokinase 1, putative
Ligand
BDBM514001
Substrate
n/a
Meas. Tech.
enzyme-inhibition screening assay
IC50
16080±160 nM
Citation
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More Info.:
Target
Name:
Glucokinase 1, putative
Synonyms:
Q4E4E1_TRYCC
Type:
Protein
Mol. Mass.:
41591.25
Organism:
Trypanosoma cruzi (strain CL Brener)
Description:
Q4E4E1
Residue:
376
Sequence:
MNIKELSLHELCEELKTPAWNVPLTFVGDVGGTSARMGFVREGKNDSVHACVTRYSMKRKDITELIEFFNEIIELMPASVIKRVKAGVINVPGPVTGGAVGGPFNNLKGIARLSDYPKALFPPGRSAILNDLEAGGFGVLAVSDAHVFSEYFGVMWEGTQWRTCEQEPAGSVIGRGRCLVLAPGTGLGSSLIYYNPMNQQHIVVPLELGSQTIPMRKDIDYIQTLHAELKLLPNYENMVSGAGLEFHYRQVVRGSRPPCSAGEIAKLASEGDANACKAMKKYHEYLMRVGSEASMALLPLTIVLVGDNIVNNAFFYRNPQNLKEMHREALNHEMERFGFQSRVTYLRQKKLLNLNLMGCYRCGLDLSVGKKQKAQL