Reaction Details Report a problem with these data
Target
Transcription activator BRG1 [1448-1575]
Ligand
BDBM394405
Substrate
n/a
Meas. Tech.
BRG1 TR-FRET Binding Assay
IC50
84.6±n/a nM
Citation
Albrecht, BK; Cote, A; Crawford, T; Duplessis, M; Good, AC; LeBlanc, Y; Magnuson, SR; Nasveschuk, CG; Romero, FA; Tang, Y; Taylor, AM Therapeutic compounds and uses thereof US Patent US10308614 Publication Date 6/4/2019
More Info.:
Target
Name:
Transcription activator BRG1 [1448-1575]
Synonyms:
ATP-dependent helicase SMARCA4 | BAF190A | BRG1 | His-BRG1 (A1448-S1575) | SMARCA4 | SMCA4_HUMAN | SNF2B | SNF2L4 | Transcription activator BRG1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
14937.42
Organism:
Homo sapiens (Human)
Description:
P51532(A1448-S1575)
Residue:
128
Sequence:
AEKLSPNPPNLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNHKYRSLNDLEKDVMLLCQNAQTFNLEGSLIYEDSIVLQSVFTSVRQKIEKEDDSEGEES