Reaction Details Report a problem with these data
Target
Protein tyrosine phosphatase type IVA 3
Ligand
BDBM50059084
Substrate
n/a
Meas. Tech.
In Vitro Biochemical Evaluation
IC50
132±3 nM
Citation
Lazo, JS; Sharlow, ER; McQueeney, KE; Wipf, P; Salamoun, JM Inhibitors of PTP4A3 for the treatment of cancer US Patent US10308663 Publication Date 6/4/2019
More Info.:
Target
Name:
Protein tyrosine phosphatase type IVA 3
Synonyms:
PRL3 | PTP4A3 | Protein-tyrosine phosphatase 4A3 | TP4A3_HUMAN
Type:
PROTEIN
Mol. Mass.:
19546.22
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1461022
Residue:
173
Sequence:
MARMNRPAPVEVSYKHMRFLITHNPTNATLSTFIEDLKKYGATTVVRVCEVTYDKTPLEKDGITVVDWPFDDGAPPPGKVVEDWLSLVKAKFCEAPGSCVAVHCVAGLGRAPVLVALALIESGMKYEDAIQFIRQKRRGAINSKQLTYLEKYRPKQRLRFKDPHTHKTRCCVM