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Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50060957
Substrate
n/a
Meas. Tech.
ChEMBL_211329 (CHEMBL818988)
IC50
12000±n/a nM
Citation
Goldbrunner, M; Loidl, G; Polossek, T; Mannschreck, A; von Angerer, E Inhibition of tubulin polymerization by 5,6-dihydroindolo[2,1-alpha]isoquinoline derivatives. J Med Chem 40:3524-33 (1997) [PubMed] Article
More Info.:
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP