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Target
Alpha-1B adrenergic receptor
Ligand
BDBM50118702
Substrate
n/a
Meas. Tech.
ChEMBL_911066 (CHEMBL3056713)
Ki
6918±n/a nM
Citation
  TBA Med Chem Res 13:134-148 (2004)    Article 
Target
Name:
Alpha-1B adrenergic receptor
Synonyms:
ADA1B_MESAU | ADRA1B | adrenergic Alpha1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
56514.13
Organism:
HAMSTER
Description:
adrenergic Alpha1 0 HAMSTER::P18841
Residue:
515
Sequence:
MNPDLDTGHNTSAPAQWGELKDANFTGPNQTSSNSTLPQLDVTRAISVGLVLGAFILFAIVGNILVILSVACNRHLRTPTNYFIVNLAIADLLLSFTVLPFSATLEVLGYWVLGRIFCDIWAAVDVLCCTASILSLCAISIDRYIGVRYSLQYPTLVTRRKAILALLSVWVLSTVISIGPLLGWKEPAPNDDKECGVTEEPFYALFSSLGSFYIPLAVILVMYCRVYIVAKRTTKNLEAGVMKEMSNSKELTLRIHSKNFHEDTLSSTKAKGHNPRSSIAVKLFKFSREKKAAKTLGIVVGMFILCWLPFFIALPLGSLFSTLKPPDAVFKVVFWLGYFNSCLNPIIYPCSSKEFKRAFMRILGCQCRSGRRRRRRRRLGACAYTYRPWTRGGSLERSQSRKDSLDDSGSCMSGSQRTLPSASPSPGYLGRGAQPPLELCAYPEWKSGALLSLPEPPGRRGRLDSGPLFTFKLLGEPESPGTEGDASNGGCDATTDLANGQPGFKSNMPLAPGHF
  
Inhibitor
Name:
BDBM50118702
Synonyms:
2-Amino-1-(2,5-dimethoxy-phenyl)-ethanol | CHEMBL1076 | DESGLYMIDODRINE | Orvaten | Proamatine
Type:
Small organic molecule
Emp. Form.:
C10H15NO3
Mol. Mass.:
197.231
SMILES:
COc1ccc(OC)c(c1)C(O)CN
Structure:
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