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Target
Histone deacetylase 2b
Ligand
BDBM50082663
Substrate
n/a
Meas. Tech.
ChEMBL_87885 (CHEMBL698803)
IC50
140±n/a nM
Citation
 Jung, M; Brosch, G; Kölle, D; Scherf, H; Gerhäuser, C; Loidl, P Amide analogues of trichostatin A as inhibitors of histone deacetylase and inducers of terminal cell differentiation. J Med Chem 42:4669-79 (1999) [PubMed]  Article 
Target
Name:
Histone deacetylase 2b
Synonyms:
Histone deacetylase HD2
Type:
PROTEIN
Mol. Mass.:
30785.07
Organism:
Zea mays
Description:
ChEMBL_87549
Residue:
286
Sequence:
MEVGGQEVKPGATVSCKVGDGLVIHLSQAALGESKKASENAILSVNIDDKKLVLGTLSVEKHPQISCDLVFDKDFELPHNSKTRSVFFRGYKSPVPLFESNSGEDSSDEELKTDQIPLQNNEIKISAAKVPAKDDDDDVFIILAMMMMIYSSDDDDDDFTTSDSDNEMSEEDDSSDEDEMSEEDDSSDEDEMSGGADPSDDSSDESGSEHTSAPKKTDVVVGKKRAIKAEAPYGKKAKSEQSSQKTGDKASTSHPAKQSIKTPADKSRKTPTADKKSPKSGSHGCK
  
Inhibitor
Name:
BDBM50082663
Synonyms:
CHEMBL143802 | N-(5-Hydroxycarbamoyl-pentyl)-4-methoxy-benzamide
Type:
Small organic molecule
Emp. Form.:
C14H20N2O4
Mol. Mass.:
280.3196
SMILES:
COc1ccc(cc1)C(=O)NCCCCCC(=O)NO
Structure:
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