Reaction Details Report a problem with these data
Target
Phospholipase A2 group V
Ligand
BDBM50262843
Substrate
n/a
Meas. Tech.
ChEMBL_489279 (CHEMBL990835)
IC50
>1600±n/a nM
Citation
Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem 51:4708-14 (2008) [PubMed] Article
More Info.:
Target
Name:
Phospholipase A2 group V
Synonyms:
PA2G5_MOUSE | Pla2g5
Type:
PROTEIN
Mol. Mass.:
15864.30
Organism:
Mus musculus
Description:
ChEMBL_700980
Residue:
137
Sequence:
MKGLLTLAWFLACSVPAVPGGLLELKSMIEKVTGKNAFKNYGFYGCYCGWGGRGTPKDGTDWCCQMHDRCYGQLEEKDCAIRTQSYDYRYTNGLVICEHDSFCPMRLCACDRKLVYCLRRNLWTYNPLYQYYPNFLC