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Target
Phosphoglycerate kinase
Ligand
BDBM50067778
Substrate
n/a
Meas. Tech.
ChEMBL_155739 (CHEMBL759844)
Kd
4000±n/a nM
Citation
Jakeman, DL; Ivory, AJ; Williamson, MP; Blackburn, GM Highly potent bisphosphonate ligands for phosphoglycerate kinase. J Med Chem 41:4439-52 (1998) [PubMed] Article
More Info.:
Target
Name:
Phosphoglycerate kinase
Synonyms:
PGK1 | PGK_YEAST | Phosphoglycerate kinase 1
Type:
PROTEIN
Mol. Mass.:
44741.88
Organism:
Saccharomyces cerevisiae
Description:
ChEMBL_155739
Residue:
416
Sequence:
MSLSSKLSVQDLDLKDKRVFIRVDFNVPLDGKKITSNQRIVAALPTIKYVLEHHPRYVVLASHLGRPNGERNEKYSLAPVAKELQSLLGKDVTFLNDCVGPEVEAAVKASAPGSVILLENLRYHIEEEGSRKVDGQKVKASKEDVQKFRHELSSLADVYINDAFGTAHRAHSSMVGFDLPQRAAGFLLEKELKYFGKALENPTRPFLAILGGAKVADKIQLIDNLLDKVDSIIIGGGMAFTFKKVLENTEIGDSIFDKAGAEIVPKLMEKAKAKGVEVVLPVDFIIADAFSADANTKTVTDKEGIPAGWQGLDNGPESRKLFAATVAKAKTIVWNGPPGVFEFEKFAAGTKALLDEVVKSSAAGNTVIIGGGDTATVAKKYGVTDKISHVSTGGGASLELLEGKELPGVAFLSEKK