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Target
P2Y purinoceptor 6
Ligand
BDBM50118239
Substrate
n/a
Meas. Tech.
ChEMBL_521733 (CHEMBL1005023)
EC50
200±n/a nM
Citation
Eliahu, SE; Camden, J; Lecka, J; Weisman, GA; Sévigny, J; Gélinas, S; Fischer, B Identification of hydrolytically stable and selective P2Y(1) receptor agonists. Eur J Med Chem 44:1525-36 (2009) [PubMed] Article
More Info.:
Target
Name:
P2Y purinoceptor 6
Synonyms:
P2RY6_RAT | P2ry6 | Pyrimidinergic receptor P2Y6
Type:
PROTEIN
Mol. Mass.:
36704.21
Organism:
Rat
Description:
ChEMBL_805344
Residue:
328
Sequence:
MERDNGTIQAPGLPPTTCVYREDFKRLLLPPVYSVVLVVGLPLNVCVIAQICASRRTLTRSAVYTLNLALADLLYACSLPLLIYNYARGDHWPFGDLACRLVRFLFYANLHGSILFLTCISFQRYLGICHPLAPWHKRGGRRAAWVVCGVVWLVVTAQCLPTAVFAATGIQRNRTVCYDLSPPILSTRYLPYGMALTVIGFLLPFTALLACYCRMARRLCRQDGPAGPVAQERRSKAARMAVVVAAVFVISFLPFHITKTAYLAVRSTPGVSCPVLETFAAAYKGTRPFASANSVLDPILFYFTQQKFRRQPHDLLQKLTAKWQRQRV