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Target
Mu-type opioid receptor
Ligand
BDBM50010483
Substrate
n/a
Meas. Tech.
ChEMBL_1353487 (CHEMBL3269823)
IC50
1.4±n/a nM
Citation
 Ballet, S; Betti, C; Novoa, A; Tömböly, C; Nielsen, CU; Helms, HC; Lesniak, A; Kleczkowska, P; Chung, NN; Lipkowski, AW; Brodin, B; Tourwé, D; Schiller, PW In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt ACS Med Chem Lett 5:352-357 (2014) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50010483
Synonyms:
CHEMBL2181202
Type:
Small organic molecule
Emp. Form.:
C32H49N9O5
Mol. Mass.:
639.7888
SMILES:
Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N[C@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(N)=O |r|
Structure:
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