Reaction Details
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Target
Equilibrative nucleoside transporter 2
Ligand
BDBM50036306
Substrate
n/a
Meas. Tech.
ChEMBL_1432011 (CHEMBL3388116)
IC50
1310±n/a nM
Citation
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More Info.:
Target
Name:
Equilibrative nucleoside transporter 2
Synonyms:
Ent2 | Equilibrative NBMPR-insensitive nucleoside transporter | Equilibrative nitrobenzylmercaptopurine riboside-insensitive nucleoside transporter | Equilibrative nucleoside transporter 2 | Nucleoside transporter, ei-type | S29A2_RAT | Slc29a2 | Solute carrier family 29 member 2
Type:
PROTEIN
Mol. Mass.:
50265.69
Organism:
Rattus norvegicus
Description:
ChEMBL_103616
Residue:
456
Sequence:
MAHGNAPRDSYHLVGISFFILGLGTLLPWNFFITAIPYFQGRLAGTNSSAETPSTNHTSPTDTFNFNNWVTLLSQLPLLLFTLLNSFLYQCIPESVRILGSLLAILLLFALTAALVKVDLSPGLFFSITMASVWFINSFCAVLQGSLFGQLGTMPSTYSTLFLSGQGLAGIFAALAMLTSLASGVDPQTSALGYFITPCVGILLSIICYLSLPHLKFARYYLTKKPQAPVQELETKAELLGADEKNGIPVSPQQAGPTLDLDPEKELELGLEEPQKPGKPSVFVVFRKIWLTALCLVLVFTVTLSVFPAITAMVTTSSNSPGKWSQFFNPICCFLLFNVMDWLGRSLTSYFLWPDEDSQLLPLLVCLRFLFVPLFMLCHVPQRARLPIIFWQDAYFITFMLLFAISNGYFVSLTMCLAPRQVLPHEREVAGALMTFFLALGLSCGASLSFLFKALL