Reaction Details Report a problem with these data
Target
D(3) dopamine receptor
Ligand
BDBM85097
Substrate
n/a
Ki
630.95±n/a nM
Comments
PDSP_1670
Citation
Kennett, GA; Wood, MD; Bright, F; Trail, B; Riley, G; Holland, V; Avenell, KY; Stean, T; Upton, N; Bromidge, S; Forbes, IT; Brown, AM; Middlemiss, DN; Blackburn, TP SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist. Neuropharmacology 36:609-20 (1997) [PubMed] Article
More Info.:
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44279.64
Organism:
Chinese hamster
Description:
DOPAMINE D3 DRD3 C.H.O.::A0A3Q0CXS4
Residue:
400
Sequence:
MAPLSQISNHINSTCGAENITGANRARPHAYYALSYCALILAIIFGNALVCAAVLRERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVQYQHGTGQSSCRRVTLMITAVWVLAFAVSCPLLFGFNTTGDPSICSISNPDFVIYSSVVSFYVPFGVTVLVYARIYMVLRQRRRKRILTRQNSQCVSIRPGFPQQPLSPGQTHGELKRYYSICQDTALRHPSFQGGGGGMSRVERTRNSLSPTMAPKLSLEVRKLSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQACHVSPELYRATTWLGYVNSALNPVIYTTFNVEFRKAFLKILSC