Reaction Details Report a problem with these data
Target
Histamine receptor H3
Ligand
BDBM22914
Substrate
n/a
Ki
6.76±n/a nM
Comments
PDSP_1847
Citation
Esbenshade, TA; Krueger, KM; Miller, TR; Kang, CH; Denny, LI; Witte, DG; Yao, BB; Fox, GB; Faghih, R; Bennani, YL; Williams, M; Hancock, AA Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects. J Pharmacol Exp Ther 305:887-96 (2003) [PubMed] Article
More Info.:
Target
Name:
Histamine receptor H3
Synonyms:
HISTAMINE H3 | HRH3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
16901.59
Organism:
Dog
Description:
Q865E3
Residue:
147
Sequence:
FLLNLAISDFLVGAFCIPLYVPYVLTGRWPFSRGLCKLWLVVDYLLCTSSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVQKMVLVWVLAFLLYGPAILSWEHLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFN