Reaction Details Report a problem with these data
Target
Trace amine-associated receptor 1
Ligand
BDBM109581
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
Ki
0.3±n/a nM
Citation
 Galley, G; Groebke Zbinden, K; Norcross, R; Stalder, H 2-aminooxazolines as TAAR1 ligands US Patent  US8604061 Publication Date 12/10/2013 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TAAR1_RAT | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1
Type:
Enzyme
Mol. Mass.:
38034.73
Organism:
Rattus norvegicus (Rat)
Description:
Q923Y9
Residue:
332
Sequence:
MHLCHNSANISHTNSNWSRDVRASLYSLISLIILTTLVGNLIVIISISHFKQLHTPTNWLLHSMAVVDFLLGCLVMPYSMVRTVEHCWYFGELFCKLHTSTDIMLSSASILHLAFISIDRYYAVCDPLRYKAKINLAAIFVMILISWSLPAVFAFGMIFLELNLEGVEELYHNQVFCLRGCFPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRANLQVGLEGESRAPQSKETKAAKTLGIMVGVFLLCWCPFFFCMVLDPFLGYVIPPTLNDTLNWFGYLNSAFNPMVYAFFYPWFRRALKMVLFGKIFQKDSSRSKLFL
  
Inhibitor
Name:
BDBM109581
Synonyms:
US8604061, 316
Type:
Small organic molecule
Emp. Form.:
C9H8BrClN2O
Mol. Mass.:
275.53
SMILES:
NC1=N[C@H](CO1)c1ccc(Br)cc1Cl |r,t:1|
Structure:
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