Reaction Details Report a problem with these data
Target
Glucose-dependent insulinotropic receptor [1-198]/[199-335]
Ligand
BDBM189335
Substrate
n/a
Meas. Tech.
Tet-Inducible cAMP Assay
EC50
3±n/a nM
Citation
Broekema, M; Wu, G; Wacker, DA Pyrimidinylpiperidinyloxypyridone analogues as GPR119 modulators US Patent US9174965 Publication Date 11/3/2015
More Info.:
Target
Name:
Glucose-dependent insulinotropic receptor [1-198]/[199-335]
Synonyms:
Human-mouse GPR119
Type:
Protein
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Glucose-dependent insulinotropic receptor [1-198]
Synonyms:
GP119_HUMAN | GPR119 | Glucose-dependent insulinotropic receptor (GPR119)
Type:
Enzyme
Mol. Mass.:
21505.57
Organism:
Homo sapiens (Human)
Description:
Q8TDV5: The first 198 amino acids of human GPR119
Residue:
198
Sequence:
MESSFSFGVILAVLASLIIATNTLVAVAVLLLIHKNDGVSLCFTLNLAVADTLIGVAISGLLTDQLSSPSRPTQKTLCSLRMAFVTSSAAASVLTVMLITFDRYLAIKQPFRYLKIMSGFVAGACIAGLWLVSYLIGFLPLGIPMFQQTAYKGQCSFFAVFHPHFVLTLSCVGFFPAMLLFVFFYCDMLKIASMHSQQ
Component 2
Name:
Glucose-dependent insulinotropic receptor [199-335]
Synonyms:
GP119_MOUSE | Glucose-dependent insulinotropic receptor (GPR119) | Gpr119
Type:
Enzyme
Mol. Mass.:
15641.79
Organism:
Mus musculus (Mouse)
Description:
Q7TQP3: C-terminal 137 amino acids of the mouse receptor GPR119
Residue:
137
Sequence:
IRKMEHAGAMAGAYRPPRSVNDFKAVRTIAVLIGSFTLSWSPFLITSIVQVACHKCCLYQVLEKYLWLLGVGNSLLNPLIYAYWQREVRQQLYHMALGVKKFFTSILLLLPARNRGPERTRESAYHIVTISHPELDG