Reaction Details Report a problem with these data
Target
Cathepsin Z
Ligand
BDBM453275
Substrate
n/a
Meas. Tech.
Inhibition of Lysine Gingipain
IC50
>10000±n/a nM
Citation
Konradi, AW; Galemmo, Jr., RA; Dominy, SS; Lynch, CC; Holsinger, LJ Ketone inhibitors of lysine gingipain US Patent US10730826 Publication Date 8/4/2020
More Info.:
Target
Name:
Cathepsin Z
Synonyms:
CATZ_HUMAN | CTSZ | Cathepsin P | Cathepsin X
Type:
PROTEIN
Mol. Mass.:
33870.59
Organism:
Human
Description:
ChEMBL_595889
Residue:
303
Sequence:
MARRGPGWRPLLLLVLLAGAAQGGLYFRRGQTCYRPLRGDGLAPLGRSTYPRPHEYLSPADLPKSWDWRNVDGVNYASITRNQHIPQYCGSCWAHASTSAMADRINIKRKGAWPSTLLSVQNVIDCGNAGSCEGGNDLSVWDYAHQHGIPDETCNNYQAKDQECDKFNQCGTCNEFKECHAIRNYTLWRVGDYGSLSGREKMMAEIYANGPISCGIMATERLANYTGGIYAEYQDTTYINHVVSVAGWGISDGTEYWIVRNSWGEPWGERGWLRIVTSTYKDGKGARYNLAIEEHCTFGDPIV