Reaction Details Report a problem with these data
Target
Tyrosine-protein kinase JAK2 [826-1132]
Ligand
BDBM458861
Substrate
n/a
Meas. Tech.
In Vitro JAK kinase Assays
IC50
0.500±n/a nM
Citation
Esteve Trias, C; Taltavull Moll, J; Gonzalez Rodriguez, J; Vidal Juan, B 2-(pyrazolopyridin-3-yl)pyrimidine derivatives as JAK inhibitors US Patent US10759793 Publication Date 9/1/2020
More Info.:
Target
Name:
Tyrosine-protein kinase JAK2 [826-1132]
Synonyms:
JAK2 | JAK2_HUMAN | Tyrosine-protein kinase JAK2 (826-1132) | Tyrosine-protein kinase JAK2 JH1 (826-1132)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
35849.63
Organism:
Human
Description:
aa 826-1132
Residue:
307
Sequence:
RIGALGFSGAFEDRDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG