Reaction Details Report a problem with these data
Target
Homeobox protein PKNOX1
Ligand
BDBM50050515
Substrate
n/a
Meas. Tech.
In Vitro Inhibition Assay
IC50
71000±n/a nM
Citation
Bachovchin, WW; Lai, H; Wu, W Combination therapies using immuno-dash inhibitors and PGE2 antagonists US Patent US11096924 Publication Date 8/24/2021
More Info.:
Target
Name:
Homeobox protein PKNOX1
Synonyms:
Homeobox protein PREP-1 | PBX/knotted homeobox 1 | PKNOX1 | PKNX1_HUMAN | PREP1
Type:
Protein
Mol. Mass.:
47590.49
Organism:
Human
Description:
P55347
Residue:
436
Sequence:
MMATQTLSIDSYQDGQQMQVVTELKTEQDPNCSEPDAEGVSPPPVESQTPMDVDKQAIYRHPLFPLLALLFEKCEQSTQGSEGTTSASFDVDIENFVRKQEKEGKPFFCEDPETDNLMVKAIQVLRIHLLELEKVNELCKDFCSRYIACLKTKMNSETLLSGEPGSPYSPVQSQQIQSAITGTISPQGIVVPASALQQGNVAMATVAGGTVYQPVTVVTPQGQVVTQTLSPGTIRIQNSQLQLQLNQDLSILHQDDGSSKNKRGVLPKHATNVMRSWLFQHIGHPYPTEDEKKQIAAQTNLTLLQVNNWFINARRRILQPMLDSSCSETPKTKKKTAQNRPVQRFWPDSIASGVAQPPPSELTMSEGAVVTITTPVNMNVDSLQSLSSDGATLAVQQVMMAGQSEDESVDSTEEDAGALAPAHISGLVLENSDSLQ