Reaction Details Report a problem with these data
Target
Bromodomain-containing protein 3 [34-140]
Ligand
BDBM528580
Substrate
n/a
Meas. Tech.
Binding Assay
IC50
35.0±n/a nM
Citation
Pham, SM; Chakravarty, S; Kankanala, J; Chen, J; Nayak, AK; Barde, A Substituted 1,6-dihydropyridinones and 1,2-dihydroisoquinolinones as bet inhibitors US Patent US11192900 Publication Date 12/7/2021
More Info.:
Target
Name:
Bromodomain-containing protein 3 [34-140]
Synonyms:
BRD3 | BRD3-1 | BRD3_HUMAN | Bromodomain-containing protein 3 (BD1, aa 34-140) | KIAA0043 | RING3L
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12880.95
Organism:
Homo sapiens (Human)
Description:
Q15059[34-140]
Residue:
107
Sequence:
RKTNQLQYMQNVVVKTLWKHQFAWPFYQPVDAIKLNLPDYHKIIKNPMDMGTIKKRLENNYYWSASECMQDFNTMFTNCYIYNKPTDDIVLMAQALEKIFLQKVAQM