Reaction Details Report a problem with these data
Target
Three-prime repair exonuclease 1
Ligand
BDBM550447
Substrate
n/a
IC50
<1000±n/a nM
Citation
Letourneau, JJ; Selvarangan Elamparuthi, K; Huang, C; Bommireddy Venkata, V Substituted pyrrolo[1,2-a]pyrazines and pyrrolo[1,2-a][1,4]diazepines as TREX1 inhibitors US Patent US11306098 Publication Date 4/19/2022
More Info.:
Target
Name:
Three-prime repair exonuclease 1
Synonyms:
3'-5' exonuclease TREX1 | TREX1_MOUSE | Trex1
Type:
Protein
Mol. Mass.:
33681.13
Organism:
Mouse
Description:
Q91XB0
Residue:
314
Sequence:
MGSQTLPHGHMQTLIFLDLEATGLPSSRPEVTELCLLAVHRRALENTSISQGHPPPVPRPPRVVDKLSLCIAPGKACSPGASEITGLSKAELEVQGRQRFDDNLAILLRAFLQRQPQPCCLVAHNGDRYDFPLLQTELARLSTPSPLDGTFCVDSIAALKALEQASSPSGNGSRKSYSLGSIYTRLYWQAPTDSHTAEGDVLTLLSICQWKPQALLQWVDEHARPFSTVKPMYGTPATTGTTNLRPHAATATTPLATANGSPSNGRSRRPKSPPPEKVPEAPSQEGLLAPLSLLTLLTLAIATLYGLFLASPGQ