Reaction Details Report a problem with these data
Target
Coagulation factor XIII B chain
Ligand
BDBM577483
Substrate
n/a
Meas. Tech.
Transamidation Assay for Determining Inhibitor Selectivity
IC50
7.00±n/a nM
Citation
Hils, M; Pasternack, R; Büchold, C Inhibitors of blood coagulation factor XIII US Patent US11472838 Publication Date 10/18/2022
More Info.:
Target
Name:
Coagulation factor XIII B chain
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
75059.25
Organism:
Rabbit
Description:
G1SEL4
Residue:
660
Sequence:
MSLKDLAFIIILIISGELHAEEKRCGFPSVENGRIAQYYYTFKSFYFPMSIDRKLPFFCLAGYTTETGKHEAQTRCTAQGWAPEPRCFKKCAKPELRNGYISDAKLAYKVRENMRYGCASGYKTTGGEDEEVVQCLADGWSSPPACRQLHETCLVPELNNGNYSTMQKTFKVKESVQYECSPGYYTAGGQKTEEVECRPHGWSVTPKCTKLKCSPLGLIEHGYFHPVKQTYEEGDVIQFFCHENYYLSGPDLIQCYNFGWYPESPVCEGRRTRCPPPPVPLNSKIQTHSTTYRHGETVHIQCELNFEIQGSEEIRCENGKWTEPPKCVEEKEKVACVQPPVIENGAANLHSETYYSGDTVSYTCESGYHLRGANEITCNRGKWTAPPECAENKEHCKPPPNVTNGAVVNESRLSYTSGSSVEYRCNEYYLLRGSKISHCEQGRWSPPPVCLEPCTVSVDDMNRNHIEMKWKYEGKVLHGDLIDFVCKRGYDISPSTPLSELSVKCNRGEVKYPLCIKKESTGMCASPPLIKHGVIIGSIVGTYENGSSIEYQCFDHYFLQGSREVYCVEGVWTTPPQCLEPCILSFFEMEKNNLRLKWDFDNRPYIFHGEYVEFLCTRNSYIAEASTLGSELRVQCVRGHLKYPRCIARESFSYQQPLQT