Reaction Details Report a problem with these data
Target
Coagulation factor XIII A chain
Ligand
BDBM577483
Substrate
n/a
Meas. Tech.
Transamidation Assay for Determining Inhibitor Selectivity
IC50
19.0±n/a nM
Citation
Hils, M; Pasternack, R; Büchold, C Inhibitors of blood coagulation factor XIII US Patent US11472838 Publication Date 10/18/2022
More Info.:
Target
Name:
Coagulation factor XIII A chain
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
82764.92
Organism:
Crab-eating macaque
Description:
A0A7N9D9X7
Residue:
728
Sequence:
MSETSRIAFGGRRAVPPNNSNAAEDDLPTLELQGVVPRGVNLQEFLNVTSIHLFKERWDTNKVDHHTDKYENNKLIVRRGQSFYIQIDFNRPYDPRRDLFRVEYVIGRYPQENKGTYIPVPIVSELQSGKWGAKIVMREDRSVRLSVQSSPECIVGKFRMYVAVWTPYGIIRTSRNPETDTYILFNPWCEDDAVYLDNEKEREEYVLNDIGVIFYGEVNDIKTRSWSYGQFEDGILDTCLYVMDRAQMDLSGRGNPIKVSRVGSAMVNAKDDEGVLVGSWDNIYAYGVPPSAWTGSVDILLEYQSSENPVRYGQCWVFAGVFNTFLRCLGIPARIVTNYFSAHDNDANLQMDIFLEEDGNVNSKLTKDSVWNYHCWNEAWMTRPDLPVGFGGWQAVDSTPQENSDGMYRCGPASVQAIKHGHVCFQFDAPFVFAEVNSDLIYITAKKDGTHVVENVDATHIGKLIVTKQIGGDGMMDITDTYKFQEERLALETALMYGAKKPLNTEGVMKSRSKVDMDFEVENAVLGKDLKLTITFRNNSHNHYTITAYLSANITFYTGVSKAEFKKETFDVTLEPLSFKKEAVLIQAGEYMGQLLEQASLHFFVTARINETSDVLAKQKSTVLTIPKLIIKVRGAQVVGSDMIVTVEFTNPLKETLRNVWIHLDGPGITRPMRKMFREIRPNSTVQWEEVCRPWVSGPRKLIASMSSDSLRHVYGELDVQIQRRPSM