Reaction Details Report a problem with these data
Target
Three-prime repair exonuclease 1
Ligand
BDBM550471
Substrate
n/a
Meas. Tech.
TREX1 Exonuclease Assay
IC50
<1000±n/a nM
Citation
Letourneau, JJ; Selvarangan Elamparuthi, K; Huang, C; Bommireddy Venkata, V Substituted pyrrolo[1,2-a]pyrazines and pyrrolo[1,2-a][1,4]diazepines as TREX1 inhibitors US Patent US11583538 Publication Date 2/21/2023
More Info.:
Target
Name:
Three-prime repair exonuclease 1
Synonyms:
3'-5' exonuclease TREX1 | DNase III | Deoxyribonuclease III | TREX1 | TREX1_HUMAN
Type:
Protein
Mol. Mass.:
33217.46
Organism:
Human
Description:
Q9NSU2
Residue:
314
Sequence:
MGSQALPPGPMQTLIFFDMEATGLPFSQPKVTELCLLAVHRCALESPPTSQGPPPTVPPPPRVVDKLSLCVAPGKACSPAASEITGLSTAVLAAHGRQCFDDNLANLLLAFLRRQPQPWCLVAHNGDRYDFPLLQAELAMLGLTSALDGAFCVDSITALKALERASSPSEHGPRKSYSLGSIYTRLYGQSPPDSHTAEGDVLALLSICQWRPQALLRWVDAHARPFGTIRPMYGVTASARTKPRPSAVTTTAHLATTRNTSPSLGESRGTKDLPPVKDPGALSREGLLAPLGLLAILTLAVATLYGLSLATPGE