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Target
ATP-sensitive inward rectifier potassium channel 10
Ligand
BDBM600745
Substrate
n/a
Meas. Tech.
thallium-flux assay
IC50
>30000±n/a nM
Citation
Swale, DR; Foil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent US11632953 Publication Date 4/25/2023
More Info.:
Target
Name:
ATP-sensitive inward rectifier potassium channel 10
Synonyms:
ATP-dependent inwardly rectifying potassium channel Kir4.1 | Inward rectifier K(+) channel Kir1.2 | KCJ10_HUMAN | KCNJ10 | Potassium channel, inwardly rectifying subfamily J member 10
Type:
PROTEIN
Mol. Mass.:
42513.64
Organism:
Homo sapiens (Human)
Description:
ChEMBL_105175
Residue:
379
Sequence:
MTSVAKVYYSQTTQTESRPLMGPGIRRRRVLTKDGRSNVRMEHIADKRFLYLKDLWTTFIDMQWRYKLLLFSATFAGTWFLFGVVWYLVAVAHGDLLELDPPANHTPCVVQVHTLTGAFLFSLESQTTIGYGFRYISEECPLAIVLLIAQLVLTTILEIFITGTFLAKIARPKKRAETIRFSQHAVVASHNGKPCLMIRVANMRKSLLIGCQVTGKLLQTHQTKEGENIRLNQVNVTFQVDTASDSPFLILPLTFYHVVDETSPLKDLPLRSGEGDFELVLILSGTVESTSATCQVRTSYLPEEILWGYEFTPAISLSASGKYIADFSLFDQVVKVASPSGLRDSTVRYGDPEKLKLEESLREQAEKEGSALSVRISNV