Reaction Details Report a problem with these data
Target
GTPase KRas [G12D]
Ligand
BDBM629382
Substrate
n/a
Meas. Tech.
Biochemical Assay
IC50
0.100±n/a nM
Citation
DAI, C; GUERRERO, JA; GUNEY, T; GUO, H; KATO, D; KIBURU, IN; LAZERWITH, SE; MCKINLEY, JL; MEDLEY, JW; PYUN, H; TIAN, M; TSUI, VH; WATKINS, WJ; ZAJDLIK, AD; ZHANG, JR KRAS G12D MODULATING COMPOUNDS US Patent US20230339981 Publication Date 10/26/2023
More Info.:
Target
Name:
GTPase KRas [G12D]
Synonyms:
GTPase KRas (G12D) | KRAS | KRAS2 | RASK2 | RASK_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
21713.12
Organism:
Homo sapiens (Human)
Description:
P01116[G12D]
Residue:
189
Sequence:
MTEYKLVVVGADGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQRVEDAFYTLVREIRQYRLKKISKEEKTPGCVKIKKCIIM