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Target
Interleukin-21
Ligand
BDBM247023
Substrate
n/a
IC50
>10000±n/a nM
Citation
 Gaweco, A; Tilley, J; Blinn, J Sulfonamide retinoic acid receptor-related orphan receptor modulators and uses thereof US Patent  US9701663 Publication Date 7/11/2017 
Target
Name:
Interleukin-21
Synonyms:
IL21 | IL21_HUMAN | Za11 | il-21
Type:
Enzyme Catalytic Domain
Mol. Mass.:
17933.60
Organism:
Homo sapiens (Human)
Description:
Q9HBE4
Residue:
162
Sequence:
MRSSPGNMERIVICLMVIFLGTLVHKSSSQGQDRHMIRMRQLIDIVDQLKNYVNDLVPEFLPAPEDVETNCEWSAFSCFQKAQLKSANTGNNERIINVSIKKLKRKPPSTNAGRRQKHRLTCPSCDSYEKKPPKEFLERFKSLLQKMIHQHLSSRTHGSEDS
  
Inhibitor
Name:
BDBM247023
Synonyms:
US9701663, 6
Type:
Small organic molecule
Emp. Form.:
C23H28N4O
Mol. Mass.:
376.4946
SMILES:
C(C1CC2CCC1N2)n1ccc2cc(ccc12)-c1cnn(c1)C1CCCCO1 |TLB:0:1:5.4:7|
Structure:
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