Reaction Details Report a problem with these data
Target
Gag-Pol polyprotein [588-1147,V662I,F664L,F703Y,Q738M,M771V]
Ligand
BDBM77092
Substrate
n/a
Meas. Tech.
PHENOSENSE assay
IC50
5.0±0.0 nM
Citation
Lanier, ER Methods of treating retroviral infections and related dosage regimes US Patent US9694024 Publication Date 7/4/2017
More Info.:
Target
Name:
Gag-Pol polyprotein [588-1147,V662I,F664L,F703Y,Q738M,M771V]
Synonyms:
HIV RT (75I/77L/116Y/151M/184V) | POL_HV1H2 | gag-pol
Type:
n/a
Mol. Mass.:
64453.42
Organism:
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Description:
P04585[588-1147,V662I,F664L,F703Y,Q738M,M771V]
Residue:
560
Sequence:
PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEGKISKIGPENPYNTPVFAIKKKDSTKWRKLIDLRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYYSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPMGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYVDDLYVGSDLEIGQHRTKIEELRQHLLRWGLTTPDKKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRKVL