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Target
Neuropeptide Y receptor type 2
Ligand
BDBM42431
Substrate
n/a
Meas. Tech.
Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism
IC50
>35000±n/a nM
Citation
 PubChem, PC Dose response counterscreen assay for neuropeptide Y receptor Y1 (NPY-Y1): Cell-based high throughput assay to measure NPY-Y2 antagonism PubChem Bioassay (2008)[AID] 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM42431
Synonyms:
MLS000589265 | N'-(2-Butyl-2-hydroxy-hexanoyl)-N-phenyl-hydrazinecarboxylic acid methyl ester | N-[(2-butyl-2-hydroxy-1-oxohexyl)amino]-N-phenylcarbamic acid methyl ester | N-[(2-butyl-2-hydroxy-hexanoyl)amino]-N-phenyl-carbamic acid methyl ester | SMR000212665 | cid_1899455 | methyl N-[(2-butyl-2-hydroxyhexanoyl)amino]-N-phenylcarbamate | methyl N-[(2-butyl-2-oxidanyl-hexanoyl)amino]-N-phenyl-carbamate
Type:
Small organic molecule
Emp. Form.:
C18H28N2O4
Mol. Mass.:
336.4259
SMILES:
CCCCC(O)(CCCC)C(=O)NN(C(=O)OC)c1ccccc1
Structure:
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