Reaction Details Report a problem with these data
Target
Protein Rev [8-24]
Ligand
BDBM44544
Substrate
n/a
Meas. Tech.
Dose response biochemical assay to identify inhibitors of the HIV Rev - RRE RNA interaction (disruption of protein-RNA interaction)
IC50
>79370±n/a nM
Citation
 PubChem, PC Dose response biochemical assay to identify inhibitors of the HIV Rev - RRE RNA interaction (disruption of protein-RNA interaction) PubChem Bioassay (2007)[AID] 
Target
Name:
Protein Rev [8-24]
Synonyms:
Chain B, Rna Aptamer Complexed With Hiv-1 Rev Peptide, Nmr, 7 Structures | REV_HV1W2 | rev
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2446.81
Organism:
Human immunodeficiency virus 1
Description:
gi_253722402
Residue:
17
Sequence:
TRQARRNRRRRWRERQR
  
Inhibitor
Name:
BDBM44544
Synonyms:
2-(4-methoxyphenyl)ethyl-[3-(4-methoxyphenyl)-1-methyl-propyl]amine | 4-(4-methoxyphenyl)-N-[2-(4-methoxyphenyl)ethyl]-2-butanamine | 4-(4-methoxyphenyl)-N-[2-(4-methoxyphenyl)ethyl]butan-2-amine | MLS000532942 | SMR000140380 | cid_2846243
Type:
Small organic molecule
Emp. Form.:
C20H27NO2
Mol. Mass.:
313.4339
SMILES:
COc1ccc(CCNC(C)CCc2ccc(OC)cc2)cc1
Structure:
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